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Partner Data
CBIS
Matrix
Example Data Type:
Secondary Screen (Kd)
Primary Screen(% control or competition)
If the input file contains Primary and Secondary Data, use:
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Assay Data File:
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Bromodomain
Kd
Primary
To highlight spots, select a compound(s), click 'fill' and select entries.
Create Images for:
Dasatinib
Highlight These Spots (
fill
):
Dasatinib|ABL1-nonphosphorylated|0.02
Dasatinib|ABL2|0.17
Dasatinib|ACVR1|620
Dasatinib|ACVR1B|330
Dasatinib|ACVR2A|210
Dasatinib|ACVR2B|570
Dasatinib|ACVRL1|460
Dasatinib|ADCK3|190
Dasatinib|AURKA|9300
Dasatinib|BLK|0.21
Dasatinib|BMPR1A|7000
Dasatinib|BMPR1B|53
Dasatinib|BMX|1.4
Dasatinib|BRAF|500
Dasatinib|BRK|7.8
Dasatinib|BTK|1.4
Dasatinib|CSF1R|0.58
Dasatinib|CSK|1
Dasatinib|CSNK1E|1500
Dasatinib|DDR1|0.69
Dasatinib|DDR2|3.2
Dasatinib|DMPK|1300
Dasatinib|DMPK2|1200
Dasatinib|EGFR|120
Dasatinib|EPHA1|4.1
Dasatinib|EPHA2|0.85
Dasatinib|EPHA3|0.09
Dasatinib|EPHA4|1.2
Dasatinib|EPHA5|0.24
Dasatinib|EPHA6|2100
Dasatinib|EPHA8|0.24
Dasatinib|EPHB1|0.45
Dasatinib|EPHB2|0.39
Dasatinib|EPHB3|6.9
Dasatinib|EPHB4|0.34
Dasatinib|EPHB6|0.03
Dasatinib|ERBB2|1400
Dasatinib|ERBB3|18
Dasatinib|ERBB4|55
Dasatinib|FGFR1|3700
Dasatinib|FGFR2|1400
Dasatinib|FGFR3|3900
Dasatinib|FGR|0.5
Dasatinib|FLT1|5000
Dasatinib|FLT3|4800
Dasatinib|FRK|0.31
Dasatinib|FYN|0.79
Dasatinib|GAK|2.6
Dasatinib|GCN2(Kin.Dom.2,S808G)|1600
Dasatinib|HCK|0.35
Dasatinib|HPK1|980
Dasatinib|JAK2(JH1domain-catalytic)|1000
Dasatinib|JAK3(JH1domain-catalytic)|640
Dasatinib|KIT|0.81
Dasatinib|LCK|0.2
Dasatinib|LIMK1|570
Dasatinib|LIMK2|86
Dasatinib|LOK|1200
Dasatinib|LYN|0.57
Dasatinib|LZK|5300
Dasatinib|MAP3K2|140
Dasatinib|MAP3K3|280
Dasatinib|MAP3K4|310
Dasatinib|MAP4K2|1300
Dasatinib|MAP4K3|640
Dasatinib|MAP4K4|3100
Dasatinib|MAP4K5|45
Dasatinib|MEK1|1000
Dasatinib|MEK2|1400
Dasatinib|MEK5|3.3
Dasatinib|MINK|430
Dasatinib|MRCKA|2000
Dasatinib|MRCKB|2100
Dasatinib|MST1|3800
Dasatinib|MST4|1900
Dasatinib|MYLK2|3500
Dasatinib|NEK11|470
Dasatinib|NEK2|6500
Dasatinib|NLK|260
Dasatinib|p38-alpha|27
Dasatinib|p38-beta|410
Dasatinib|PDGFRA|0.47
Dasatinib|PDGFRB|0.63
Dasatinib|PKMYT1|130
Dasatinib|QSK|28
Dasatinib|RAF1|570
Dasatinib|RET|730
Dasatinib|RIPK2|31
Dasatinib|SBK1|1200
Dasatinib|SIK|3.9
Dasatinib|SIK2|6.4
Dasatinib|SLK|720
Dasatinib|SRC|0.21
Dasatinib|SRMS|13
Dasatinib|STK35|770
Dasatinib|STK36|210
Dasatinib|SYK|2900
Dasatinib|TAK1|3700
Dasatinib|TAOK2|5400
Dasatinib|TAOK3|2300
Dasatinib|TEC|13
Dasatinib|TESK1|33
Dasatinib|TGFBR1|230
Dasatinib|TGFBR2|2900
Dasatinib|TNIK|2000
Dasatinib|TNK2|5.6
Dasatinib|TNNI3K|11
Dasatinib|TXK|2.1
Dasatinib|TYK2(JH1domain-catalytic)|1800
Dasatinib|TYK2(JH2domain-pseudokinase)|110
Dasatinib|ULK3|4600
Dasatinib|VEGFR2|2900
Dasatinib|VRK2|3200
Dasatinib|WEE1|7000
Dasatinib|WEE2|200
Dasatinib|YES|0.3
Dasatinib|YSK1|3400
Dasatinib|YSK4|79
Dasatinib|ZAK|45
Dasatinib|ABL1-nonphosphorylated
Dasatinib|ABL2
Dasatinib|ACVR1
Dasatinib|ACVR1B
Dasatinib|ACVR2A
Dasatinib|ACVR2B
Dasatinib|ACVRL1
Dasatinib|ADCK3
Dasatinib|AURKA
Dasatinib|BLK
Dasatinib|BMPR1A
Dasatinib|BMPR1B
Dasatinib|BMX
Dasatinib|BRAF
Dasatinib|BRK
Dasatinib|BTK
Dasatinib|CSF1R
Dasatinib|CSK
Dasatinib|CSNK1E
Dasatinib|DDR1
Dasatinib|DDR2
Dasatinib|DMPK
Dasatinib|DMPK2
Dasatinib|EGFR
Dasatinib|EPHA1
Dasatinib|EPHA2
Dasatinib|EPHA3
Dasatinib|EPHA4
Dasatinib|EPHA5
Dasatinib|EPHA6
Dasatinib|EPHA8
Dasatinib|EPHB1
Dasatinib|EPHB2
Dasatinib|EPHB3
Dasatinib|EPHB4
Dasatinib|EPHB6
Dasatinib|ERBB2
Dasatinib|ERBB3
Dasatinib|ERBB4
Dasatinib|FGFR1
Dasatinib|FGFR2
Dasatinib|FGFR3
Dasatinib|FGR
Dasatinib|FLT1
Dasatinib|FLT3
Dasatinib|FRK
Dasatinib|FYN
Dasatinib|GAK
Dasatinib|GCN2(Kin.Dom.2,S808G)
Dasatinib|HCK
Dasatinib|HPK1
Dasatinib|JAK2(JH1domain-catalytic)
Dasatinib|JAK3(JH1domain-catalytic)
Dasatinib|KIT
Dasatinib|LCK
Dasatinib|LIMK1
Dasatinib|LIMK2
Dasatinib|LOK
Dasatinib|LYN
Dasatinib|LZK
Dasatinib|MAP3K2
Dasatinib|MAP3K3
Dasatinib|MAP3K4
Dasatinib|MAP4K2
Dasatinib|MAP4K3
Dasatinib|MAP4K4
Dasatinib|MAP4K5
Dasatinib|MEK1
Dasatinib|MEK2
Dasatinib|MEK5
Dasatinib|MINK
Dasatinib|MRCKA
Dasatinib|MRCKB
Dasatinib|MST1
Dasatinib|MST4
Dasatinib|MYLK2
Dasatinib|NEK11
Dasatinib|NEK2
Dasatinib|NLK
Dasatinib|p38-alpha
Dasatinib|p38-beta
Dasatinib|PDGFRA
Dasatinib|PDGFRB
Dasatinib|PKMYT1
Dasatinib|QSK
Dasatinib|RAF1
Dasatinib|RET
Dasatinib|RIPK2
Dasatinib|SBK1
Dasatinib|SIK
Dasatinib|SIK2
Dasatinib|SLK
Dasatinib|SRC
Dasatinib|SRMS
Dasatinib|STK35
Dasatinib|STK36
Dasatinib|SYK
Dasatinib|TAK1
Dasatinib|TAOK2
Dasatinib|TAOK3
Dasatinib|TEC
Dasatinib|TESK1
Dasatinib|TGFBR1
Dasatinib|TGFBR2
Dasatinib|TNIK
Dasatinib|TNK2
Dasatinib|TNNI3K
Dasatinib|TXK
Dasatinib|TYK2(JH1domain-catalytic)
Dasatinib|TYK2(JH2domain-pseudokinase)
Dasatinib|ULK3
Dasatinib|VEGFR2
Dasatinib|VRK2
Dasatinib|WEE1
Dasatinib|WEE2
Dasatinib|YES
Dasatinib|YSK1
Dasatinib|YSK4
Dasatinib|ZAK
Dasatinib|ABL1-nonphosphorylated|0.02
Dasatinib|ABL2|0.17
Dasatinib|ACVR1|620
Dasatinib|ACVR1B|330
Dasatinib|ACVR2A|210
Dasatinib|ACVR2B|570
Dasatinib|ACVRL1|460
Dasatinib|ADCK3|190
Dasatinib|AURKA|9300
Dasatinib|BLK|0.21
Dasatinib|BMPR1A|7000
Dasatinib|BMPR1B|53
Dasatinib|BMX|1.4
Dasatinib|BRAF|500
Dasatinib|BRK|7.8
Dasatinib|BTK|1.4
Dasatinib|CSF1R|0.58
Dasatinib|CSK|1
Dasatinib|CSNK1E|1500
Dasatinib|DDR1|0.69
Dasatinib|DDR2|3.2
Dasatinib|DMPK|1300
Dasatinib|DMPK2|1200
Dasatinib|EGFR|120
Dasatinib|EPHA1|4.1
Dasatinib|EPHA2|0.85
Dasatinib|EPHA3|0.09
Dasatinib|EPHA4|1.2
Dasatinib|EPHA5|0.24
Dasatinib|EPHA6|2100
Dasatinib|EPHA8|0.24
Dasatinib|EPHB1|0.45
Dasatinib|EPHB2|0.39
Dasatinib|EPHB3|6.9
Dasatinib|EPHB4|0.34
Dasatinib|EPHB6|0.03
Dasatinib|ERBB2|1400
Dasatinib|ERBB3|18
Dasatinib|ERBB4|55
Dasatinib|FGFR1|3700
Dasatinib|FGFR2|1400
Dasatinib|FGFR3|3900
Dasatinib|FGR|0.5
Dasatinib|FLT1|5000
Dasatinib|FLT3|4800
Dasatinib|FRK|0.31
Dasatinib|FYN|0.79
Dasatinib|GAK|2.6
Dasatinib|GCN2(Kin.Dom.2,S808G)|1600
Dasatinib|HCK|0.35
Dasatinib|HPK1|980
Dasatinib|JAK2(JH1domain-catalytic)|1000
Dasatinib|JAK3(JH1domain-catalytic)|640
Dasatinib|KIT|0.81
Dasatinib|LCK|0.2
Dasatinib|LIMK1|570
Dasatinib|LIMK2|86
Dasatinib|LOK|1200
Dasatinib|LYN|0.57
Dasatinib|LZK|5300
Dasatinib|MAP3K2|140
Dasatinib|MAP3K3|280
Dasatinib|MAP3K4|310
Dasatinib|MAP4K2|1300
Dasatinib|MAP4K3|640
Dasatinib|MAP4K4|3100
Dasatinib|MAP4K5|45
Dasatinib|MEK1|1000
Dasatinib|MEK2|1400
Dasatinib|MEK5|3.3
Dasatinib|MINK|430
Dasatinib|MRCKA|2000
Dasatinib|MRCKB|2100
Dasatinib|MST1|3800
Dasatinib|MST4|1900
Dasatinib|MYLK2|3500
Dasatinib|NEK11|470
Dasatinib|NEK2|6500
Dasatinib|NLK|260
Dasatinib|p38-alpha|27
Dasatinib|p38-beta|410
Dasatinib|PDGFRA|0.47
Dasatinib|PDGFRB|0.63
Dasatinib|PKMYT1|130
Dasatinib|QSK|28
Dasatinib|RAF1|570
Dasatinib|RET|730
Dasatinib|RIPK2|31
Dasatinib|SBK1|1200
Dasatinib|SIK|3.9
Dasatinib|SIK2|6.4
Dasatinib|SLK|720
Dasatinib|SRC|0.21
Dasatinib|SRMS|13
Dasatinib|STK35|770
Dasatinib|STK36|210
Dasatinib|SYK|2900
Dasatinib|TAK1|3700
Dasatinib|TAOK2|5400
Dasatinib|TAOK3|2300
Dasatinib|TEC|13
Dasatinib|TESK1|33
Dasatinib|TGFBR1|230
Dasatinib|TGFBR2|2900
Dasatinib|TNIK|2000
Dasatinib|TNK2|5.6
Dasatinib|TNNI3K|11
Dasatinib|TXK|2.1
Dasatinib|TYK2(JH1domain-catalytic)|1800
Dasatinib|TYK2(JH2domain-pseudokinase)|110
Dasatinib|ULK3|4600
Dasatinib|VEGFR2|2900
Dasatinib|VRK2|3200
Dasatinib|WEE1|7000
Dasatinib|WEE2|200
Dasatinib|YES|0.3
Dasatinib|YSK1|3400
Dasatinib|YSK4|79
Dasatinib|ZAK|45
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Dasatinib
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Dasatinib
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* WildType kinase assays appear in both the main TREEspot and Mutant kinase dendrogams.
Human Kinome image created by KINOMEscan.
2 images created. To download (copy and paste) all images to your local machine click Open/Browse Image Folder.
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Dasatinib
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